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PEPA
CAS No. 141286-78-4
PEPA( —— )
Catalog No. M26365 CAS No. 141286-78-4
PEPA is an allosteric AMPA receptors modulator; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 32 | In Stock |
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| 5MG | 30 | In Stock |
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| 10MG | 46 | In Stock |
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| 25MG | 101 | In Stock |
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| 50MG | 193 | In Stock |
|
| 100MG | 287 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePEPA
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NoteResearch use only, not for human use.
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Brief DescriptionPEPA is an allosteric AMPA receptors modulator; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity.
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DescriptionPEPA is an allosteric AMPA receptors modulator; binds to the GluA2o and GluA3o LBDs and can be utilized as an indicator of AMPA receptor heterogeneity.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetiGluR
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RecptorPDE4
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Research Area——
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Indication——
Chemical Information
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CAS Number141286-78-4
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Formula Weight402.43
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Molecular FormulaC16H16F2N2O4S2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (124.24 mM)
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SMILESNC(=O)COc1c(F)cc(SCCNS(=O)(=O)c2ccccc2)cc1F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zhao Y, Zhang HT, O'Donnell JM. Inhibitor binding to type 4 phosphodiesterase (PDE4) assessed using [3H]piclamilast and [3H]rolipram. J Pharmacol Exp Ther. 2003 May;305(2):565-72. doi: 10.1124/jpet.102.47407. Erratum in: J Pharmacol Exp Ther. 2003 Dec;307(3):1243.
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