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Home - Products - Angiogenesis - c-Met/HGFR - Hepln-13

Hepln-13

CAS No. 64369-13-7

Hepln-13( Hepln 13 | Hepln13 )

Catalog No. M24659 CAS No. 64369-13-7

Hepln-13 is a hepsin inhibitor that acts by hindering prostate cancer bone metastasis.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 84 In Stock
2MG 44 In Stock
5MG 73 In Stock
10MG 122 In Stock
25MG 244 In Stock
50MG 356 In Stock
100MG 496 In Stock
200MG 685 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock
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Biological Information

  • Product Name
    Hepln-13
  • Note
    Research use only, not for human use.
  • Brief Description
    Hepln-13 is a hepsin inhibitor that acts by hindering prostate cancer bone metastasis.
  • Description
    Hepln-13 is a hepsin inhibitor that acts by hindering prostate cancer bone metastasis.
  • In Vitro
    Hepln-13 (10 μM; 2 hours; 293 cells) inhibits cleavage.Western Blot Analysis Cell Line:293 cells Concentration:10 μM Incubation Time:2 hours Result:Inhibited cleavage.
  • In Vivo
    HepIn-13 displays dose dependent inhibition of Hepsin overexpression-relevant prostate cancer phenotypes and blocks prostate cancer metastasis.
  • Synonyms
    Hepln 13 | Hepln13
  • Pathway
    Angiogenesis
  • Target
    c-Met/HGFR
  • Recptor
    hepsin
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    64369-13-7
  • Formula Weight
    325.2
  • Molecular Formula
    C17H13BrN2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:60 mg/mL?(184.50 mM;?Need ultrasonic)
  • SMILES
    Brc1ccc(C(N2)Nc3cccc4cccc2c34)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Tang X, et al. Targeted inhibition of cell-surface serine protease Hepsin blocks prostate cancer bone metastasis. Oncotarget. 2014;5(5):1352-1362.
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