Tacrine

CAS No. 321-64-2

Tacrine( CS 12602 | Tacrinum )

Catalog No. M24254 CAS No. 321-64-2

Tacrine is an indirect cholinergic agonist and centrally acting anticholinesterase.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 33 In Stock
5MG 29 In Stock
10MG 46 In Stock
25MG 92 In Stock
50MG 129 In Stock
100MG 183 In Stock
200MG Get Quote In Stock
500MG 368 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Tacrine
  • Note
    Research use only, not for human use.
  • Brief Description
    Tacrine is an indirect cholinergic agonist and centrally acting anticholinesterase.
  • Description
    Tacrine is an indirect cholinergic agonist and centrally acting anticholinesterase. It is approved for the treatment of Alzheimer's disease.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    CS 12602 | Tacrinum
  • Pathway
    Endocrinology/Hormones
  • Target
    AChR
  • Recptor
    Cholinergic
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    321-64-2
  • Formula Weight
    198.26
  • Molecular Formula
    C13H14N2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:Soluble; Water:Insoluble
  • SMILES
    Nc1c(CCCC2)c2nc2ccccc12
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ismaili L, Refouvelet B, Benchekroun M, Brogi S, Brindisi M, Gemma S, Campiani G, Filipic S, Agbaba D, Esteban G, Unzeta M, Nikolic K, Butini S, Marco-Contelles J. Multitarget compounds bearing tacrine- and donepezil-like structural and functional motifs for the potential treatment of Alzheimer's disease. Prog Neurobiol. 2016 Jan 18. pii: S0301-0082(15)00162-8. doi: 10.1016/j.pneurobio.2015.12.003. [Epub ahead of print] Review.
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