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(Rac)-JBJ-04-125-02
CAS No. 2140807-05-0
(Rac)-JBJ-04-125-02( —— )
Catalog No. M23974 CAS No. 2140807-05-0
JBJ-04-125-02 is effective as a single agent in both in vitro and in vivo models of EGFR-mutant lung cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 262 | In Stock |
|
| 5MG | 217 | In Stock |
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| 10MG | 353 | In Stock |
|
| 25MG | 598 | In Stock |
|
| 50MG | 833 | In Stock |
|
| 100MG | 1135 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product Name(Rac)-JBJ-04-125-02
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NoteResearch use only, not for human use.
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Brief DescriptionJBJ-04-125-02 is effective as a single agent in both in vitro and in vivo models of EGFR-mutant lung cancer.
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DescriptionJBJ-04-125-02 is effective as a single agent in both in vitro and in vivo models of EGFR-mutant lung cancer.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetEGFR
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RecptorEGFR (L858R/T790M )
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Research Area——
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Indication——
Chemical Information
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CAS Number2140807-05-0
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Formula Weight543.6
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Molecular FormulaC29H26FN5O3S
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Purity>98% (HPLC)
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SolubilityDMSO:240mg/mL (441.5 mM);Water:Insoluble
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SMILESC1CN(CCN1)C2=CC=C(C=C2)C3=CC4=C(CN(C4=O)C(C5=C(C=CC(=C5)F)O)C(=O)NC6=NC=CS6)C=C3
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Single and Dual Targeting of Mutant EGFR with an Allosteric Inhibitor
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