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HPK1-IN-2
CAS No. 2056122-11-1
HPK1-IN-2( Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-HPK1-IN-2 )
Catalog No. M23923 CAS No. 2056122-11-1
HPK1-IN-2 is a potent and orally active inhibitor of hematopoietic progenitor kinase-1 (HPK1;IC50<0.05 μΜ).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 164 | In Stock |
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| 5MG | 139 | In Stock |
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| 10MG | 231 | In Stock |
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| 25MG | 386 | In Stock |
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| 50MG | 537 | In Stock |
|
| 100MG | 714 | In Stock |
|
| 200MG | 918 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameHPK1-IN-2
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NoteResearch use only, not for human use.
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Brief DescriptionHPK1-IN-2 is a potent and orally active inhibitor of hematopoietic progenitor kinase-1 (HPK1;IC50<0.05 μΜ).
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DescriptionHPK1-IN-2 is a potent and orally active inhibitor of hematopoietic progenitor kinase-1 (HPK1;IC50<0.05 μΜ). It also inhibits Lck (0.05 μΜIn Vitro——In Vivo——SynonymsThieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-HPK1-IN-2PathwayAngiogenesisTargetFLTRecptorFlt3|HPK1|LckResearch Area——Indication——
Chemical Information
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CAS Number2056122-11-1
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Formula Weight380.47
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Molecular FormulaC19H20N6OS
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Purity>98% (HPLC)
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SolubilityH2O:25 mg/mL?(55.14 mM;?Need ultrasonic)
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SMILESO=C1C(C2=NC3=CC=C(N4CCN(C)CC4)C=C3N2)=C(N)C(C=CS5)=C5N1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Peter Brent Sampson, et al. Hpk1 inhibitors and methods of using same. WO2016205942A1.
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