CD38 inhibitor 1( —— )

Catalog No. M23764 CAS No. 1700637-55-3

CD38 inhibitor 1 is an inhibitor of CD38. For hCD38 and mouse CD38, the IC50s are 7.3 nM and 1.9 nM.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

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Biological Information

Product Name

CD38 inhibitor 1
Note

Research use only, not for human use.
Brief Description

CD38 inhibitor 1 is an inhibitor of CD38. For hCD38 and mouse CD38, the IC50s are 7.3 nM and 1.9 nM.
Description

CD38 inhibitor 1 is an inhibitor of CD38. For hCD38 and mouse CD38, the IC50s are 7.3 nM and 1.9 nM.
In Vitro

——
In Vivo

CD38 inhibitor (30 mg/kg; oral administration; 2 and 6 hours) significantly elevates NAD levels in liver and muscle. Animal Model:Diet induced obese (DIO) C57Bl6 miceDosage:30 mg/kg Administration:Orally onceResult:NAD levels were significantly increased at both the 2 and 6 h time points in liver and muscle.
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

CD38
Research Area

——
Indication

——

Chemical Information

CAS Number

1700637-55-3
Formula Weight

413.53
Molecular Formula

C22H27N3O3S
Purity

>98% (HPLC)
Solubility

DMSO:35.71 mg/mL (86.35 mM; Need ultrasonic)
SMILES

CN(c(ccc(-c1cncs1)c1)c1C(NC(CC1)CCC1OCCOC)=C1)C1=O
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Haffner CD, et al. Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors. J Med Chem. 2015 Apr 23;58(8):3548-71.

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