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HIF-2α-IN-2
CAS No. 1672666-82-8
HIF-2α-IN-2( —— )
Catalog No. M23751 CAS No. 1672666-82-8
HIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 101 | In Stock |
|
| 5MG | 91 | In Stock |
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| 10MG | 125 | In Stock |
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| 25MG | 217 | In Stock |
|
| 50MG | 306 | In Stock |
|
| 100MG | 425 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameHIF-2α-IN-2
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NoteResearch use only, not for human use.
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Brief DescriptionHIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).
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DescriptionHIF-2α-IN-2 is a hypoxia-inducible factor (HIF-2α) inhibitor (IC50: 16 nM in scintillation proximity assay).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetHIF/HIF Prolyl-hydroxylase
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RecptorHIF-2α
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Research Area——
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Indication——
Chemical Information
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CAS Number1672666-82-8
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Formula Weight365.35
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Molecular FormulaC17H13F2NO4S
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Purity>98% (HPLC)
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SolubilityDMSO:100 mg/mL (273.71 mM; Need ultrasonic)
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SMILESN#CC1=CC(OC2=CC=C(S(=O)(C)=O)C3=C2CC(F)C3O)=CC(F)=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Darryl David DIXON, et al. Aryl ethers and uses thereof. WO2015035223A1.
molnova catalog
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HIF2α-IN-2
HIF2α-IN-2 is a potent, selective, allosteric inhibitor of HIF-2α PAS-B domain with Kd of 81 nM.
