Sofpironium bromide

CAS No. 1628106-94-4

Sofpironium bromide( BBI-4000 | BBI4000 | BBI 4000 )

Catalog No. M23722 CAS No. 1628106-94-4

Sofpironium bromide belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 160 In Stock
5MG 155 In Stock
10MG 250 In Stock
25MG 452 In Stock
50MG 665 In Stock
100MG 986 In Stock
200MG 1321 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Sofpironium bromide
  • Note
    Research use only, not for human use.
  • Brief Description
    Sofpironium bromide belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.
  • Description
    Sofpironium bromide belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.
  • In Vitro
    Sofpironium bromide is metabolized mainly through non-enzymatic hydrolysis, and also through oxidative metabolism via CYP2D6 and CYP3A4.
  • In Vivo
    Sofpironium bromide exhibits anticholinergic activity by inhibiting the contractile activity of guinea pig ileal tissue in a concentration-dependent manner. In a rat model, Sofpironium bromide reduces footpad sweating induced by Pilocarpine (a muscarinic receptor agonist).
  • Synonyms
    BBI-4000 | BBI4000 | BBI 4000
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    others
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1628106-94-4
  • Formula Weight
    470.4
  • Molecular Formula
    C22H32BrNO5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:95 mg/mL?(201.95 mM;?Need ultrasonic)
  • SMILES
    CCOC(C[N+](C)(CC1)C[C@@H]1OC([C@@](C2CCCC2)(C3=CC=CC=C3)O)=O)=O.[Br-]
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Julia Paik, et al. Sofpironium Bromide: First Approval. Drugs. 2020 Dec;80(18):1981-1986.
molnova catalog
related products
  • JNJ-65355394

    JNJ-65355394 is an effective O-GlcNAc hydrolase (OGA) inhibitor and an OGA chemical probe.

  • MAO-IN-M30 dihydroch...

    Potent and brain selective monoamine oxidase (MAO) inhibitor (EC50 values are 37 and 57 nM for MAO-A and MAO-B, respectively).

  • 2-Hydroxy-1-Methoxya...

    2-Hydroxy-1-Methoxyaporphine can inhibit CYP2D6 activity, it also increase the glucose consumption significantly as rosiglitazone.