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Home - Products - GPCR/G Protein - Dopamine Receptor - GR 103691

GR 103691

CAS No. 162408-66-4

GR 103691( —— )

Catalog No. M23720 CAS No. 162408-66-4

GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 55 In Stock
10MG 91 In Stock
25MG 186 In Stock
50MG 295 In Stock
100MG 478 In Stock
500MG 1062 In Stock
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Biological Information

  • Product Name
    GR 103691
  • Note
    Research use only, not for human use.
  • Brief Description
    GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).
  • Description
    GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM). It shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 and hD1 sites.
  • In Vitro
    GR 103691 shows marked affinity for serotonin1A (5-HT1A) receptors (Ki of 5.8 nM) and α-1 adrenoceptors (Ki of 12.6 nM).
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Dopamine Receptor
  • Recptor
    D3
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    162408-66-4
  • Formula Weight
    485.62
  • Molecular Formula
    C30H35N3O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:10 mM
  • SMILES
    O=C(C1=CC=C(C2=CC=C(C(C)=O)C=C2)C=C1)NCCCCN3CCN(C4=CC=CC=C4OC)CC3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Audinot V, et al. A comparative in vitro and in vivo pharmacological characterization of the novel dopamine D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194. J Pharmacol Exp Ther. 1998 Oct;287(1):187-97.
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