Seralutinib

CAS No. 1619931-27-9

Seralutinib( GB002 )

Catalog No. M23717 CAS No. 1619931-27-9

Seralutinib is an inhibitor of inhaled PDGFRα and PDGFRβ. It is used in the study for pulmonary arterial hypertension.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 93 In Stock
2MG 56 In Stock
5MG 93 In Stock
10MG 140 In Stock
25MG 250 In Stock
50MG 323 In Stock
100MG 514 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Seralutinib
  • Note
    Research use only, not for human use.
  • Brief Description
    Seralutinib is an inhibitor of inhaled PDGFRα and PDGFRβ. It is used in the study for pulmonary arterial hypertension.
  • Description
    Seralutinib is an inhibitor of inhaled PDGFRα and PDGFRβ. It is used in the study for pulmonary arterial hypertension.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    GB002
  • Pathway
    Angiogenesis
  • Target
    PDGFR
  • Recptor
    PDGFRα|PDGFRβ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1619931-27-9
  • Formula Weight
    469.55
  • Molecular Formula
    C27H27N5O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:100 mg/mL?(212.98 mM;?Need ultrasonic)
  • SMILES
    CC1=CC(=CN=C1)C(=O)NC2=CC=CC(=C2)[C@H](C)NC3=NC(=CN=C3)C4=CC(=C(C=C4)OC)OC
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Anna Galkin, et al. Pharmacologic Characterization of GB002, a Novel Inhaled PDGFR Kinase Inhibitor in Development for Pulmonary Arterial Hypertension (PAH).
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