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Tesmilifene fumarate

CAS No. 1185241-83-1

Tesmilifene fumarate( DPPE fumarate )

Catalog No. M23352 CAS No. 1185241-83-1

Tesmilifene fumarate (DPPE fumarate) is an H1C receptor antagonist。

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Tesmilifene fumarate
  • Note
    Research use only, not for human use.
  • Brief Description
    Tesmilifene fumarate (DPPE fumarate) is an H1C receptor antagonist。
  • Description
    Tesmilifene fumarate (DPPE fumarate) is an H1C receptor antagonist。
  • In Vitro
    Tesmilifene may modulate the effects of 12(S)HETE in cancer cells, and indirectly, influence the susceptibility of cellular DNA to chemotherapy.
  • In Vivo
    Tesmilifene (DPPE, 20 mg/kg (s.c.) and 20 μg (icv in 5 μL)) potentiated seizures induced by both convulsants. Animal Model:Male BKTO mice (25-45 g).Dosage:20 mg/kg (s.c.) and 20 μg (icv in 5 μL).Administration:S.C. and icv.Result:Potentiated seizures induced by both convulsants.
  • Synonyms
    DPPE fumarate
  • Pathway
    GPCR/G Protein
  • Target
    Histamine Receptor
  • Recptor
    Histamine Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1185241-83-1
  • Formula Weight
    399.48
  • Molecular Formula
    C23H29NO5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:248 mg/mL (620.81 mM; Need ultrasonic)
  • SMILES
    CCN(CC)CCOC1=CC=C(C=C1)CC2=CC=CC=C2.OC(/C=C/C(O)=O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Mark Vincent, et al. Tesmilifene may enhance breast cancer chemotherapy by killing a clone of aggressive, multi-drug resistant cells through its action on the p-glycoprotein pump. Med Hypotheses. 2006;66(4):715-31.
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