CIM0216

CAS No. 1031496-06-6

CIM0216( N-(5-methyl-1,2-oxazol-3-yl)-2-phenyl-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide )

Catalog No. M23235 CAS No. 1031496-06-6

CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 88 In Stock
2MG 51 In Stock
5MG 80 In Stock
10MG 141 In Stock
25MG 297 In Stock
50MG 456 In Stock
100MG 686 In Stock
200MG Get Quote In Stock
500MG 1423 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CIM0216
  • Note
    Research use only, not for human use.
  • Brief Description
    CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.
  • Description
    CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    N-(5-methyl-1,2-oxazol-3-yl)-2-phenyl-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    TRP/TRPV Channel
  • Recptor
    TRPM3
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1031496-06-6
  • Formula Weight
    347.41
  • Molecular Formula
    C21H21N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 30 mg/mL?(86.35 mM;?Need ultrasonic and warming);Ethanol: 17 mg/mL?(48.93 mM;?Need ultrasonic and warming)
  • SMILES
    O=C(NC1=NOC(C)=C1)C(C2=CC=CC=C2)N3CCCC4=C3C=CC=C4
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Vriens J , Owsianik G , Hofmann T , et al. TRPM3 is a nociceptor channel involved in the detection of noxious heat.[J]. Neuron, 2011, 70(3):482-494.
molnova catalog
related products
  • SN 2

    SN 2 is a novel and potent TRPML3 ion channel activator(EC50 = 1.13 μM). SN 2 also shares a similar antiviral effect against DENV2 and ZIKV.

  • TC-I 2014

    TC-I 2014 shows antiallodynic properties in pain models.

  • JNJ-38893777 sulfate

    JNJ-38893777 is a potent and selective transient receptor potential vanilloid 1 (TRPV1) channel antagonist for treatment of ociceptive and neuropathic pain.