PF-06882961( —— )

Catalog No. M22917 CAS No. 2230198-02-2

COA

Datasheet

HNMR

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MSDS

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Product Name

PF-06882961
Note

Research use only, not for human use.
Brief Description

PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist. PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat.
Description

PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist. PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat.
In Vitro

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In Vivo

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Synonyms

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Pathway

GPCR/G Protein
Target

Glucagon Receptor
Recptor

GLP-1
Research Area

Metabolism
Indication

Diabetes Mellitus, Type 2

CAS Number

2230198-02-2
Formula Weight

555.6
Molecular Formula

C31H30FN5O4
Purity

>98% (HPLC)
Solubility

DMSO:125 mg/mL (224.98 mM; Need ultrasonic)
SMILES

OC(C1=CC=C(N=C(CN2CCC(C3=NC(OCC4=CC=C(C#N)C=C4F)=CC=C3)CC2)N5C[C@H]6OCC6)C5=C1)=O
Chemical Name

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