GABAA receptor agent 1

CAS No. 1571-87-5

GABAA receptor agent 1( —— )

Catalog No. M22616 CAS No. 1571-87-5

GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 79 In Stock
5MG 72 In Stock
10MG 113 In Stock
25MG 226 In Stock
50MG 333 In Stock
100MG 485 In Stock
200MG 668 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    GABAA receptor agent 1
  • Note
    Research use only, not for human use.
  • Brief Description
    GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.
  • Description
    GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.
  • In Vitro
    ——
  • In Vivo
    GABAA receptor agent 1 (30 mg/kg; intraperitoneal) inhibits the maximum electroshock (MES) and pentylenetetrazole (PTZ)-induced convulsions in swiss albino rats.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GABAA
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1571-87-5
  • Formula Weight
    273.67
  • Molecular Formula
    C13H8ClN3O2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 83.33 mg/mL (304.49 mM)
  • SMILES
    [O-][N+](=O)c1ccc2nc([nH]c2c1)-c1ccc(Cl)cc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Jain P, et al. Design, synthesis and biological evaluation of some novel benzimidazole derivatives for their potential anticonvulsant activity. Arch Pharm Res. 2010 Jul;33(7):971-80.
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