Taltirelin acetate

CAS No. 1549593-23-8

Taltirelin acetate( TA-0910 acetate )

Catalog No. M22365 CAS No. 1549593-23-8

Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 49 In Stock
2MG 29 In Stock
5MG 45 In Stock
10MG 73 In Stock
25MG 144 In Stock
50MG 237 In Stock
100MG 369 In Stock
200MG 547 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Taltirelin acetate
  • Note
    Research use only, not for human use.
  • Brief Description
    Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).
  • Description
    Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    TA-0910 acetate
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    THR
  • Research Area
    Nervous system
  • Indication
    Spinocerebellar Degeneration

Chemical Information

  • CAS Number
    1549593-23-8
  • Formula Weight
    465.46
  • Molecular Formula
    C19H27N7O7
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL (268.55 mM; Need ultrasonic)
  • SMILES
    O=C(N(CCC1)[C@@H]1C(N)=O)[C@@H](NC([C@@H](NC2=O)CC(N2C)=O)=O)CC3=CN=CN3.CC(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne). 2012 Oct 9;3:120.
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