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Vorolanib
CAS No. 1013920-15-4
Vorolanib( CM082,X-82 )
Catalog No. M21932 CAS No. 1013920-15-4
Vorolanib is an orally active VEGFR/PDGFR dual inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 250 | In Stock |
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| 2MG | 145 | In Stock |
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| 5MG | 227 | In Stock |
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| 10MG | 359 | In Stock |
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| 25MG | 616 | In Stock |
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| 50MG | 870 | In Stock |
|
| 100MG | 1181 | In Stock |
|
| 200MG | 1572 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameVorolanib
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NoteResearch use only, not for human use.
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Brief DescriptionVorolanib is an orally active VEGFR/PDGFR dual inhibitor.
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DescriptionVorolanib is an orally active VEGFR/PDGFR dual inhibitor.
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In Vitro——
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In Vivo——
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SynonymsCM082,X-82
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PathwayAngiogenesis
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TargetVEGFR
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RecptorVEGFR|PDGFR
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Research AreaUrinary system/Cancer
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IndicationRenal Cell Cancer Metastatic
Chemical Information
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CAS Number1013920-15-4
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Formula Weight439.48
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Molecular FormulaC23H26FN5O3
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Purity>98% (HPLC)
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SolubilityDMSO:22 mg/ml (50.06 mM; Need ultrasonic)
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SMILESCN(C)C(=O)N1CC[C@@H](C1)NC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Bendell JC, et al. Phase I, First-in-Human, Dose-Escalation Study to Evaluate the Safety, Tolerability, and Pharmacokinetics of Vorolanib in Patients with Advanced Solid Tumors. Oncologist. 2019 Apr;24(4):455-e121.
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