XP-59

CAS No. 890402-73-0

XP-59( —— )

Catalog No. M21756 CAS No. 890402-73-0

XP-59 is a potent inhibitor of the SARS-CoV Mpro, with a Ki of 0.1 μM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 76 In Stock
5MG 69 In Stock
10MG 113 In Stock
25MG 201 In Stock
50MG 300 In Stock
100MG 417 In Stock
200MG 589 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    XP-59
  • Note
    Research use only, not for human use.
  • Brief Description
    XP-59 is a potent inhibitor of the SARS-CoV Mpro, with a Ki of 0.1 μM.
  • Description
    XP-59 is a potent inhibitor of the SARS-CoV Mpro, with a Ki of 0.1 μM.
  • In Vitro
    The SARS-CoV main proteinase (Mpro) plays a central role in the formation of the viral replicase/transcriptase complex and is thus an ideal target for the development of suitable drugs.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    890402-73-0
  • Formula Weight
    282.3
  • Molecular Formula
    C??H??N?O?
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : 62.5 mg/mL (221.40 mM; Need ultrasonic)
  • SMILES
    O=C(ON1N=NC2=CC=CC=C21)C3=CC=C(N(C)C)C=C3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Verschueren KH, et al,. A structural view of the inactivation of the SARS coronavirus main proteinase by benzotriazole esters. Chem Biol. 2008 Jun;15(6):597-606.
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