YM976

CAS No. 191219-80-4

YM976( —— )

Catalog No. M21141 CAS No. 191219-80-4

YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 51 In Stock
5MG 41 In Stock
10MG 67 In Stock
25MG 110 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    YM976
  • Note
    Research use only, not for human use.
  • Brief Description
    YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM).
  • Description
    YM976 is an orally active PDE4 inhibitor (IC50:2.2 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    PDE
  • Recptor
    PDE4
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    191219-80-4
  • Formula Weight
    313.78
  • Molecular Formula
    C17H16ClN3O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CCc1ccc2c(-c3cccc(Cl)c3)nc(=O)n(CC)c2n1
  • Chemical Name
    4-(3-chlorophenyl)-17-diethyl-1H2H-pyrido[23-d]pyrimidin-2-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Aoki M Kobayashi M Ishikawa J et al. A Novel Phosphodiesterase Type 4 Inhibitor YM976 (4-(3-Chlorophenyl)-17-diethylpyrido[23-d]pyrimidin-2(1H)-one) with Little Emetogenic Activity[J]. Journal of Pharmacology & Experimental Therapeutics 2000 295(1):255-260.
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