Dermorphin TFA

CAS No. 78331-26-7

Dermorphin TFA( —— )

Catalog No. M21054 CAS No. 78331-26-7

Dermorphin TFA is a new class of opioids-like peptides.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 136 In Stock
5MG 187 In Stock
10MG 283 In Stock
25MG 527 In Stock
50MG 742 In Stock
100MG 1014 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Dermorphin TFA
  • Note
    Research use only, not for human use.
  • Brief Description
    Dermorphin TFA is a new class of opioids-like peptides.
  • Description
    Dermorphin TFA is a new class of opioids-like peptides.
  • In Vitro
    Dermorphin, a peptide isolated from the skin of Phyllomedusa frogs and the peptide receptor (NOP) component by the endogenous agonist nociceptin/orphanin FQ (N/OFQ). In displacement binding studies at CHOhMu, Dermorphin and DeNo displac the binding of [3H]-DPN in a concentration dependent and saturable manner. Dermorphin displays an affinity of 7.17, while N/OFQ fails to displace [3H]-DPN at the Delta receptor. Dermorphin and DeNo stimulate the binding of GTPγ[35S] in a concentration dependent and saturable manner at the Mu receptor.
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Others
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    78331-26-7
  • Formula Weight
    916.89
  • Molecular Formula
    C42H51F3N8O12
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C[C@@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CO)C(N)=O.O=C(O)C(F)(F)F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Castiglione R D Faoro F Perseo G et al. SYNTHESIS OF DERMORPHINS A NEW CLASS OF OPIATE-LIKE PEPTIDES[J]. Chemical Biology & Drug Design 1981 17(2):263-272.
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