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Elagolix sodium
CAS No. 832720-36-2
Elagolix sodium( NBI-56418 sodium )
Catalog No. M20990 CAS No. 832720-36-2
Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM respectively).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 65 | In Stock |
|
| 2MG | 29 | In Stock |
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| 5MG | 46 | In Stock |
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| 10MG | 69 | In Stock |
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| 25MG | 140 | In Stock |
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| 50MG | 222 | In Stock |
|
| 100MG | 352 | In Stock |
|
| 200MG | 520 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameElagolix sodium
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NoteResearch use only, not for human use.
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Brief DescriptionElagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM respectively).
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DescriptionElagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM respectively).
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In Vitro——
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In Vivo——
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SynonymsNBI-56418 sodium
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PathwayOthers
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TargetOther Targets
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RecptorGNRHR
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Research AreaCancer
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IndicationUterine leiomyoma
Chemical Information
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CAS Number832720-36-2
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Formula Weight653.57
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Molecular FormulaC32H29F5N3NaO5
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Purity>98% (HPLC)
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SolubilityDMSO:50 mg/mL (76.50 mM); H2O:50 mg/mL (76.50 mM)
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SMILESCOc1cccc(-c2c(C)n(Cc3c(F)cccc3C(F)(F)F)c(=O)n(CC(NCCCC(=O)[O-])c3ccccc3)c2=O)c1F.[Na+]
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Barra F Scala C Ferrero S2.Elagolix sodium for the treatment of women with moderate to severe endometriosis-associated pain.Drugs Today (Barc). 2019 Apr;55(4):237-246.
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