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R1487
CAS No. 449811-92-1
R1487( —— )
Catalog No. M20961 CAS No. 449811-92-1
R1487 is an orally bioavailable and highly selective p38α mitogen-activated protein kinase inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 268 | Get Quote |
|
| 10MG | 408 | Get Quote |
|
| 25MG | 672 | Get Quote |
|
| 50MG | 945 | Get Quote |
|
| 100MG | 1278 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameR1487
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NoteResearch use only, not for human use.
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Brief DescriptionR1487 is an orally bioavailable and highly selective p38α mitogen-activated protein kinase inhibitor.
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DescriptionR1487 is an orally bioavailable and highly selective p38α mitogen-activated protein kinase inhibitor.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMAPK/ERK Signaling
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Targetp38 MAPK
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Recptorp38α
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Research Area——
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Indication——
Chemical Information
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CAS Number449811-92-1
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Formula Weight388.36
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Molecular FormulaC19H18F2N4O3
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Purity>98% (HPLC)
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Solubility——
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SMILESCn1c(=O)c(Oc2ccc(F)cc2F)cc2cnc(NC3CCOCC3)nc21
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Dunford E C Herbst E A Jeoung N H et al. PDH activation during in vitro muscle contractions in PDH kinase 2 knockout mice: Effect of PDH kinase 1 compensation[J]. American Journal of Physiology Regulatory Integrative & Comparative Physiology 2011 300(6):R1487.
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