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Y15
CAS No. 4506-66-5
Y15( 1245-Benzenetetramine tetrahydrochlor | FAK inhibitor Y15 | FAK Inhibitor 14 )
Catalog No. M20681 CAS No. 4506-66-5
Y15 is a potent and specificsmall-molecule FAK scaffolding inhibitor that inhibits its autophosphorylation activity blocks tumor growth.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 38 | In Stock |
|
| 10MG | 41 | In Stock |
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| 25MG | 60 | In Stock |
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| 50MG | 70 | In Stock |
|
| 100MG | 129 | In Stock |
|
| 200MG | 184 | In Stock |
|
| 500MG | 325 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameY15
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NoteResearch use only, not for human use.
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Brief DescriptionY15 is a potent and specificsmall-molecule FAK scaffolding inhibitor that inhibits its autophosphorylation activity blocks tumor growth.
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DescriptionY15 is a potent and specificsmall-molecule FAK scaffolding inhibitor that inhibits its autophosphorylation activity blocks tumor growth.
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In Vitro——
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In Vivo——
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Synonyms1245-Benzenetetramine tetrahydrochlor | FAK inhibitor Y15 | FAK Inhibitor 14
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PathwayAngiogenesis
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TargetFAK
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RecptorFAK
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Research Area——
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Indication——
Chemical Information
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CAS Number4506-66-5
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Formula Weight284.01
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Molecular FormulaC6H14Cl4N4
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Purity>98% (HPLC)
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SolubilityH2O:59 mg/mL (207.74 mM; Need ultrasonic and warming)
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SMILESCl.Cl.Cl.Cl.Nc1cc(N)c(N)cc1N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.O'Brien S Golubovskaya VM Conroy Jet al.FAK inhibition with small molecule inhibitor Y15 decreases viability clonogenicity and cell attachment in thyroid cancer cell lines and synergizes with targeted therapeutics[J].Oncotarget. 2014 Sep 15;5(17):7945-59.
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