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PROTAC ERRα ligand 2
CAS No. 2306388-57-6
PROTAC ERRα ligand 2( —— )
Catalog No. M20565 CAS No. 2306388-57-6
PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 92 | In Stock |
|
| 5MG | 84 | In Stock |
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| 10MG | 112 | In Stock |
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| 25MG | 199 | In Stock |
|
| 50MG | 293 | In Stock |
|
| 100MG | 439 | In Stock |
|
| 200MG | 613 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePROTAC ERRα ligand 2
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NoteResearch use only, not for human use.
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Brief DescriptionPROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
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DescriptionPROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptorERRα
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Research Area——
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Indication——
Chemical Information
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CAS Number2306388-57-6
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Formula Weight445.31
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Molecular FormulaC20H13F6NO4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 62.5 mg/mL (140.35 mM)
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SMILESCOc1cc(\C=C(/C#N)C(O)=O)ccc1OCc1ccc(cc1C(F)(F)F)C(F)(F)F
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Peng L Zhang Z Lei C et al. Identification of New Small-Molecule Inducers of Estrogen-Related Receptor alpha (ERRa) Degradation[J]. ACS Medicinal Chemistry Letters 2019 10(5).
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