PROTAC ERRα ligand 2

CAS No. 2306388-57-6

PROTAC ERRα ligand 2( —— )

Catalog No. M20565 CAS No. 2306388-57-6

PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 79 In Stock
5MG 132 In Stock
10MG 177 In Stock
25MG 356 In Stock
50MG 537 In Stock
100MG 767 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    PROTAC ERRα ligand 2
  • Note
    Research use only, not for human use.
  • Brief Description
    PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
  • Description
    PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    Estrogen Receptor/ERR
  • Recptor
    ERRα
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2306388-57-6
  • Formula Weight
    445.31
  • Molecular Formula
    C20H13F6NO4
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 62.5 mg/mL (140.35 mM)
  • SMILES
    COc1cc(\C=C(/C#N)C(O)=O)ccc1OCc1ccc(cc1C(F)(F)F)C(F)(F)F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Peng L Zhang Z Lei C et al. Identification of New Small-Molecule Inducers of Estrogen-Related Receptor alpha (ERRa) Degradation[J]. ACS Medicinal Chemistry Letters 2019 10(5).
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