Fluralaner

CAS No. 864731-61-3

Fluralaner( AH252723 | A1443 )

Catalog No. M20104 CAS No. 864731-61-3

Fluralaner is an isoxazoline ectoparasiticide. It potently and selectively inhibits binding of the GABA receptor channel blocker EBOB to housefly head membranes (IC50: 455 pM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 28 In Stock
10MG 29 In Stock
25MG 56 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Fluralaner
  • Note
    Research use only, not for human use.
  • Brief Description
    Fluralaner is an isoxazoline ectoparasiticide. It potently and selectively inhibits binding of the GABA receptor channel blocker EBOB to housefly head membranes (IC50: 455 pM).
  • Description
    Fluralaner is an isoxazoline ectoparasiticide. It potently and selectively inhibits binding of the GABA receptor channel blocker EBOB to housefly head membranes (IC50: 455 pM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    AH252723 | A1443
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GABA
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    864731-61-3
  • Formula Weight
    556.29
  • Molecular Formula
    C22H17Cl2F6N3O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 100 mg/mL (179.76 mM);Water: Insoluble
  • SMILES
    Cc1cc(ccc1C(=O)NCC(=O)NCC(F)(F)F)C1=NOC(C1)(c1cc(Cl)cc(Cl)c1)C(F)(F)F
  • Chemical Name
    4-(5-(35-dichlorophenyl)-5-(trifluoromethyl)-45-dihydroisoxazol-3-yl)-2-methyl-N-(2-oxo-2-((222-trifluoroethyl)amino)ethyl)benzamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Ozoe Y et al. The antiparasitic isoxazoline A1443 is a potent blocker of insect ligand-gated chloride channels. Biochem Biophys Res Commun. 2010 Jan 1;391(1):744-9.
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