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Zacopride hydrochloride
CAS No. 101303-98-4
Zacopride hydrochloride( —— )
Catalog No. M20083 CAS No. 101303-98-4
Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 72 | In Stock |
|
| 5MG | 65 | In Stock |
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| 10MG | 101 | In Stock |
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| 25MG | 223 | In Stock |
|
| 50MG | 398 | In Stock |
|
| 100MG | 639 | In Stock |
|
| 200MG | 888 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameZacopride hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionZacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
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DescriptionZacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT3 antagonist| 5-HT4 agonist| IK1/Kir2.1 agonist
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Research Area——
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Indication——
Chemical Information
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CAS Number101303-98-4
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Formula Weight346.26
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Molecular FormulaC15H20ClN3O2.HCl
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Purity>98% (HPLC)
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SolubilityDMSO:10 mM
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SMILESCl.COc1cc(N)c(Cl)cc1C(=O)NC1CN2CCC1CC2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Nagakura Y et al. Pharmacological properties of a novel gastrointestinal prokinetic benzamide selective for human 5-HT4 receptor versus human 5-HT3 receptor. Pharmacol Res. 1999 May;39(5):375-82.
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