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PQ401 hydrochloride
CAS No. ——
PQ401 hydrochloride( —— )
Catalog No. M19402 CAS No. ——
PQ401 inhibits autophosphorylation of IGF-1R domain with IC50 of <1 μM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 49 | Get Quote |
|
| 5MG | 74 | Get Quote |
|
| 10MG | 104 | Get Quote |
|
| 25MG | 184 | Get Quote |
|
| 50MG | 331 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePQ401 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionPQ401 inhibits autophosphorylation of IGF-1R domain with IC50 of <1 μM.
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DescriptionPQ401 inhibits autophosphorylation of IGF-1R domain with IC50 of <1 μM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetIGF-1R
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RecptorIGF-1R
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Research AreaCancer
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IndicationCancer
Chemical Information
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CAS Number——
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Formula Weight378.25
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Molecular FormulaC18H17Cl2N3O2
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Purity>98% (HPLC)
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SolubilityDMSO:10 mM
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SMILESCl.COc1ccc(Cl)cc1NC(=O)Nc1cc(C)nc2ccccc12
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Gable KLetal Diarylureas are small-molecule inhibitors of insulin-like growth factor I receptor signaling and breast cancer cell growth. Mol Cancer Ther. 2006 Apr;5(4):1079-86.
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