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Pitofenone hydrochloride
CAS No. 1248-42-6
Pitofenone hydrochloride( Pitofenone hydrochloride | Pitofenone HCl | Bulgarketone )
Catalog No. M17905 CAS No. 1248-42-6
Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 28 | In Stock |
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| 10MG | 41 | In Stock |
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| 25MG | 93 | In Stock |
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| 50MG | 174 | In Stock |
|
| 100MG | 327 | In Stock |
|
| 200MG | 458 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePitofenone hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionPitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.
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DescriptionPitofenone hydrochloride is an antispasmodic agent. It acts as a potent inhibitor of acetylcholinesterase activity.
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In Vitro——
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In Vivo——
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SynonymsPitofenone hydrochloride | Pitofenone HCl | Bulgarketone
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PathwayOthers
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TargetOther Targets
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RecptorAChE
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Research Area——
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Indication——
Chemical Information
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CAS Number1248-42-6
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Formula Weight403.9
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Molecular FormulaC22H26ClNO4
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Purity>98% (HPLC)
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SolubilityDMSO : 103.3 mg/mL 255.76 mM;
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SMILESCl.O=C(OC)c1ccccc1C(=O)c3ccc(OCCN2CCCCC2)cc3
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Chemical NameMethyl 2-[4-(2-piperidin-1-ylethoxy)benzoyl]benzoate hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Punekar NS,etal.Acetylcholinesterase inhibition by pitofenone: a spasmolytic compound.Biotechnol Appl Biochem. 1991 Dec;14(3):378-82.
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