(S/R)-Orteronel

CAS No. 426219-18-3

(S/R)-Orteronel( —— )

Catalog No. M17508 CAS No. 426219-18-3

TAK-700 (Orteronel) is a potent and highly selective human 17, 20-lyase inhibitor with IC50 of 38 nM, exhibits >1000-fold selectivity over other CYPs (e.g. 11-hydroxylase and CYP3A4). Phase 3.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 85 In Stock
2MG 46 In Stock
5MG 76 In Stock
10MG 132 In Stock
25MG 264 In Stock
50MG 416 In Stock
100MG 601 In Stock
200MG 826 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    (S/R)-Orteronel
  • Note
    Research use only, not for human use.
  • Brief Description
    TAK-700 (Orteronel) is a potent and highly selective human 17, 20-lyase inhibitor with IC50 of 38 nM, exhibits >1000-fold selectivity over other CYPs (e.g. 11-hydroxylase and CYP3A4). Phase 3.
  • Description
    TAK-700 (Orteronel) is a potent and highly selective human 17, 20-lyase inhibitor with IC50 of 38 nM, exhibits >1000-fold selectivity over other CYPs (e.g. 11-hydroxylase and CYP3A4). Phase 3.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    17,20-lyase (Human) , 17,20-lyase (Rat)
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    426219-18-3
  • Formula Weight
    307.35
  • Molecular Formula
    C18H17N3O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CNC(=O)C1=CC2=C(C=C1)C=C(C=C2)C3(CCN4C3=CN=C4)O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Kaku T, et al. Bioorg Med Chem. 2011, 19(21), 6383-6399.
molnova catalog
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