Home - Products - Endocrinology/Hormones - Estrogen Receptor/ERR - L-778123 hydrochloride

L-778123 hydrochloride

CAS No. 253863-00-2

L-778123 hydrochloride( L-778,123 hydrochloride )

Catalog No. M17457 CAS No. 253863-00-2

The L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	60	In Stock
2MG	36	In Stock
5MG	58	In Stock
10MG	85	In Stock
25MG	151	In Stock
50MG	244	In Stock
100MG	411	In Stock
200MG	Get Quote	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

Get Quotation Bulk Inquiry Add to Cart

Biological Information

Product Name

L-778123 hydrochloride
Note

Research use only, not for human use.
Brief Description

The L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.
Description

The L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.
In Vitro

——
In Vivo

——
Synonyms

L-778,123 hydrochloride
Pathway

Endocrinology/Hormones
Target

Estrogen Receptor/ERR
Recptor

Farnesyl transferase (FTase)
Research Area

Cancer
Indication

——

Chemical Information

CAS Number

253863-00-2
Formula Weight

442.34
Molecular Formula

C22H21Cl2N5O
Purity

>98% (HPLC)
Solubility

DMSO : ≥ 25 mg/mL; 56.52 mM
SMILES

c1cc(cc(c1)N1CCN(Cc2cncn2Cc2ccc(cc2)C#N)CC1=O)Cl.Cl
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Lobell RB, et al. Mol Y Ther. 2002 Jul;1(9):747-58.

Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog

related products

Estrogen receptor mo...

Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active and selective estrogen receptor modulator (SERM) (pIC50: 0.46).
Droloxifene

A nonsteroidal selective estrogen receptor modulator (SERM) that shows 10- to 60-fold increased affinity for the estrogen receptor compared with Tamoxifen.
Ethynodiol diacetate

Ethynodiol diacetate is one of the first synthetic progestogens used in contraceptive pills.

Sign In Join Free