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L-778123 hydrochloride
CAS No. 253863-00-2
L-778123 hydrochloride( L-778,123 hydrochloride )
Catalog No. M17457 CAS No. 253863-00-2
The L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 60 | In Stock |
|
| 2MG | 36 | In Stock |
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| 5MG | 58 | In Stock |
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| 10MG | 85 | In Stock |
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| 25MG | 151 | In Stock |
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| 50MG | 244 | In Stock |
|
| 100MG | 411 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameL-778123 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionThe L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.
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DescriptionThe L-778123 hydrochloride is an inhibitor of FPTase (IC50: 2 nM) and GGPTase-I (IC50: 98 nM) in enzyme inhibition determination.
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In Vitro——
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In Vivo——
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SynonymsL-778,123 hydrochloride
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PathwayEndocrinology/Hormones
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TargetEstrogen Receptor/ERR
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RecptorFarnesyl transferase (FTase)
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number253863-00-2
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Formula Weight442.34
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Molecular FormulaC22H21Cl2N5O
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Purity>98% (HPLC)
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SolubilityDMSO : ≥ 25 mg/mL; 56.52 mM
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SMILESc1cc(cc(c1)N1CCN(Cc2cncn2Cc2ccc(cc2)C#N)CC1=O)Cl.Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Lobell RB, et al. Mol Y Ther. 2002 Jul;1(9):747-58.
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