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Src Inhibitor 1
CAS No. 179248-59-0
Src Inhibitor 1( Src I1 | Src I-1 | SrcI1 )
Catalog No. M17379 CAS No. 179248-59-0
Src Inhibitor 1 is a potent and selective dual site Src tyrosine kinase inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 51 | In Stock |
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| 2MG | 32 | In Stock |
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| 5MG | 51 | In Stock |
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| 10MG | 86 | In Stock |
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| 25MG | 176 | In Stock |
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| 50MG | 276 | In Stock |
|
| 100MG | 444 | In Stock |
|
| 200MG | 635 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSrc Inhibitor 1
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NoteResearch use only, not for human use.
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Brief DescriptionSrc Inhibitor 1 is a potent and selective dual site Src tyrosine kinase inhibitor.
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DescriptionSrc I1 is a potent, competitive dual site (ATP- and peptide-binding) Src kinase inhibitor (IC50 values are 44 and 88 nM for Src and Lck respectively).
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In Vitro——
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In Vivo——
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SynonymsSrc I1 | Src I-1 | SrcI1
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PathwayImmunology/Inflammation
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TargetLipoxygenase
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RecptorLck| Src
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number179248-59-0
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Formula Weight373.4
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Molecular FormulaC22H19N3O3
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Purity>98% (HPLC)
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SolubilityDMSO : 9.09 mg/mL. 24.34 mM;
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SMILESCOc1c(cc2c(c1)c(ncn2)Nc1ccc(cc1)Oc1ccccc1)OC
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Chemical Name6,7-Dimethoxy-N-(4-phenoxyphenyl)-4-quinazolinamine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Tian G, et al. Structural determinants for potent, selective dual site inhibition of human pp60c-src by 4-anilinoquinazolines. Biochemistry. 2001 Jun 19;40(24):7084-91.
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