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Saclofen
CAS No. 125464-42-8
Saclofen( Saclofen )
Catalog No. M17221 CAS No. 125464-42-8
Saclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 110 | In Stock |
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| 5MG | 116 | In Stock |
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| 10MG | 187 | In Stock |
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| 25MG | 359 | In Stock |
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| 50MG | 569 | In Stock |
|
| 100MG | 889 | In Stock |
|
| 200MG | 1200 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSaclofen
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NoteResearch use only, not for human use.
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Brief DescriptionSaclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM).
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DescriptionSaclofen is a sulfonic analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA) that acts as a competitive antagonist of the GABAB receptor (IC50: 7.8 μM). This compound can be used to determine the functional roles for the GABAB receptor as a mediator of slow inhibitory postsynaptic potentials in the brain.
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In Vitro——
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In Vivo——
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SynonymsSaclofen
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PathwayEndocrinology/Hormones
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TargetAndrogen Receptor (AR)
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RecptorGABAB
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Research Area——
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Indication——
Chemical Information
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CAS Number125464-42-8
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Formula Weight249.71
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Molecular FormulaC9H12ClNO3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?H2O : 10 mg/mL (40.05 mM)
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SMILESNCC(CS(O)(=O)=O)c1ccc(Cl)cc1
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Chemical Name3-Amino-2-(4-chlorophenyl)propane-1-sulfonic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Drew C A, Johnston G A R, Kerr D I B, et al. Neuroscience letters, 1990, 113(1): 107-110.
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