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Home - Products - Cell Cycle/DNA Damage - PARP - Desmethyl-VS-5584

Desmethyl-VS-5584

CAS No. 1246535-95-4

Desmethyl-VS-5584( Desmethyl-VS-5584 | Desmethyl-VS5584 )

Catalog No. M17217 CAS No. 1246535-95-4

Desmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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10MG 243 In Stock
25MG 408 In Stock
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Biological Information

  • Product Name
    Desmethyl-VS-5584
  • Note
    Research use only, not for human use.
  • Brief Description
    Desmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
  • Description
    Desmethyl-VS-5584 is a demethyl analogue of VS-5584, which is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Desmethyl-VS-5584 | Desmethyl-VS5584
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    PARP
  • Recptor
    mTOR| PI3K
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1246535-95-4
  • Formula Weight
    340.39
  • Molecular Formula
    C16H20N8O
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Nc1ncc(c2c3ncn(C(C)C)c3nc(N3CCOCC3)n2)cn1
  • Chemical Name
    5-[9-(1-Methylethyl)-2-(4-morpholinyl)-9H-purin-6-yl]-2-pyrimidinamine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Shao Z,et al. VS-5584, a Novel PI3K-mTOR Dual Inhibitor, Inhibits Melanoma Cell Growth In Vitro and In Vivo. PLoS One. 2015 Jul 23;10(7).
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