Endoxifen E-isomer hydrochloride

CAS No. 1197194-61-8

Endoxifen E-isomer hydrochloride( E-Endoxifen hydrochloride )

Catalog No. M17183 CAS No. 1197194-61-8

Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 182 In Stock
5MG 202 In Stock
10MG 299 In Stock
100MG Get Quote In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Endoxifen E-isomer hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
  • Description
    Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
  • In Vitro
    Endoxifen E-isomer (1-1000 nM; 12 h) inhibits PGR gene expression in E2-induced MCF-7 cells.
  • In Vivo
    ——
  • Synonyms
    E-Endoxifen hydrochloride
  • Pathway
    Proteasome/Ubiquitin
  • Target
    Tyrosinase
  • Recptor
    ERR
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1197194-61-8
  • Formula Weight
    409.95
  • Molecular Formula
    C25H28ClNO2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : ≥ 30 mg/mL. 73.18 mM
  • SMILES
    CC/C(=C(/c1ccc(cc1)O)\c1ccc(cc1)OCCNC)/c1ccccc1.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Chae YJ, et al. Eur J Pharmacol. 2015 Apr 5;752:1-7.
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