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PI3K inhibitor X
CAS No. 956958-53-5
PI3K inhibitor X( XL-147 analog )
Catalog No. M16833 CAS No. 956958-53-5
PI3K inhibitor X (XL-147 analog) is a derivative of XL147 that acts as a reversible inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 85 | In Stock |
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| 2MG | 30 | In Stock |
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| 5MG | 48 | In Stock |
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| 10MG | 76 | In Stock |
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| 25MG | 135 | In Stock |
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| 50MG | 212 | In Stock |
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| 100MG | 365 | In Stock |
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| 200MG | 475 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NamePI3K inhibitor X
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NoteResearch use only, not for human use.
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Brief DescriptionPI3K inhibitor X (XL-147 analog) is a derivative of XL147 that acts as a reversible inhibitor.
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DescriptionPI3K inhibitor X (XL-147 analog) is a derivative of XL147 that acts as a reversible inhibitor of class I PI3Ks with IC50 of 39, 36, 23 and 383 nM for p110α, δ, γ and β respectively; Compound 147 in patent WO2012006552A1.
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In Vitro——
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In Vivo——
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SynonymsXL-147 analog
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorDNA-PK|PI3Kα|PI3Kβ|PI3Kγ|PI3Kδ
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number956958-53-5
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Formula Weight448.5208
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Molecular FormulaC21H16N6O2S2
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=S(C1=CC=C(C)C=C1)(NC2=NC3=CC=CC=C3N=C2NC4=CC5=NSN=C5C=C4)=O
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Chemical NameBenzenesulfonamide, N-[3-(2,1,3-benzothiadiazol-5-ylamino)-2-quinoxalinyl]-4-methyl-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Carlos L. Arteaga, et al. Combinations of kinase inhibitors for the treatment of cancer. WO 2012006552 A1.
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