Lorediplon

CAS No. 917393-39-6

Lorediplon( GF-015535-00 )

Catalog No. M16588 CAS No. 917393-39-6

A partial positive allosteric GABAA receptor modulator.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 41 In Stock
10MG 37 In Stock
25MG 76 In Stock
50MG 144 In Stock
100MG 226 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Lorediplon
  • Note
    Research use only, not for human use.
  • Brief Description
    A partial positive allosteric GABAA receptor modulator.
  • Description
    A partial positive allosteric GABAA receptor modulator; displays activity at the alpha1-subunit, associated with promoting sleep.Sleep Disorder Phase 1 Clinical.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    GF-015535-00
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    GAT
  • Recptor
    GAT
  • Research Area
    Neurological Disease
  • Indication
    Sleep Disorder

Chemical Information

  • CAS Number
    917393-39-6
  • Formula Weight
    394.4221
  • Molecular Formula
    C20H15FN4O2S
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    CC(N(C1=CC(C2=CC=NC3=C(C(C4=CC=CS4)=O)C=NN23)=CC=C1F)C)=O
  • Chemical Name
    Acetamide, N-[2-fluoro-5-[3-(2-thienylcarbonyl)pyrazolo[1,5-a]pyrimidin-7-yl]phenyl]-N-methyl-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Zisapel N. Expert Opin Investig Drugs. 2015 Mar;24(3):401-11.
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