Brexpiprazole

CAS No. 913611-97-9

Brexpiprazole( OPC 34712 )

Catalog No. M16564 CAS No. 913611-97-9

Brexpiprazole is a novel D2 dopamine partial agonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 48 In Stock
5MG 43 In Stock
10MG 58 In Stock
25MG 69 In Stock
50MG 79 In Stock
100MG 94 In Stock
200MG 140 In Stock
500MG 268 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Brexpiprazole
  • Note
    Research use only, not for human use.
  • Brief Description
    Brexpiprazole is a novel D2 dopamine partial agonist.
  • Description
    Brexpiprazole is a novel D2 dopamine partial agonist.
  • In Vitro
    ——
  • In Vivo
    Animal Model:Male C57BL/6NCrSlc mice, Dizocilpine (0.1 mg/kg) (HY-15084B) induced social recognition deficits Dosage:0.01, 0.03 and 0.1 mg/kg Administration:Oral administration, once Result:Significantly ameliorated Dizocilpine-induced social recognition deficits, without sedation or a reduction of exploratory behavior.
  • Synonyms
    OPC 34712
  • Pathway
    Endocrinology/Hormones
  • Target
    5-HT Receptor
  • Recptor
    5-HT1A| 5-HT2A| α1B-adrenergic receptor| α2C receptors| D2L
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    913611-97-9
  • Formula Weight
    433.57
  • Molecular Formula
    C25H27N3O2S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 10 mM
  • SMILES
    O=C1NC2=C(C=C1)C=CC(OCCCCN1CCN(CC1)C1=C3C=CSC3=CC=C1)=C2
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Zajdel P, et al. Future Med Chem, 2014. 6(1): p. 57-75.
molnova catalog
related products
  • Ondansetron hydrochl...

    Ondansetron is a serotonin 5-HT receptor antagonist used mainly as anantiemetic (to treat nausea and vomiting), often following chemotherapy.

  • Homoeriodictyol

    Homoeriodictyol, a naturally occurring, bitter-masking flavanone, as a promising agent to increase appetite and food intake. The flavanone homoeriodictyol can increase SGLT-1-mediated glucose uptake but decrease serotonin release in differentiated Caco-2 cells.In contrast to other polyphenols, the flavanon Homoeriodictyol promotes glucose uptake by 29.0 ± 3.83% at a concentration of 100 μM.

  • cis-Urocanic acid

    cis-Urocanic acid is a 5-HT2A receptor agonist (Kd: 4.6 nM). It is an immune modulator that induces immunosuppression by binding to the 5-HT2A receptor.