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Setiptiline maleate

CAS No. 85650-57-3

Setiptiline maleate( MO-8282 )

Catalog No. M16210 CAS No. 85650-57-3

A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 47 In Stock
10MG 47 In Stock
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Biological Information

  • Product Name
    Setiptiline maleate
  • Note
    Research use only, not for human use.
  • Brief Description
    A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist.
  • Description
    A tetracyclic antidepressant (TeCA) that acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, as well as an H1 receptor inverse agonist/antihistamine.Depression Approved.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MO-8282
  • Pathway
    GPCR/G Protein
  • Target
    5-HT Receptor
  • Recptor
    5-HT Receptor
  • Research Area
    Neurological Disease
  • Indication
    Depression

Chemical Information

  • CAS Number
    85650-57-3
  • Formula Weight
    377.433
  • Molecular Formula
    C23H23NO4
  • Purity
    >98% (HPLC)
  • Solubility
    10 mM in DMSO
  • SMILES
    CN1CCC2=C(C1)C3=CC=CC=C3CC4=CC=CC=C24.C(=CC(=O)O)C(=O)O
  • Chemical Name
    1H-Dibenzo[3,4:6,7]cyclohepta[1,2-c]pyridine, 2,3,4,9-tetrahydro-2-methyl-, (2Z)-2-butenedioate (1:1)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Niho T, et al. Nihon Yakurigaku Zasshi. 1986 Oct;88(4):309-20. 2. Mizota M, et al. Nihon Yakurigaku Zasshi. 1986 Dec;88(6):457-66. 3. Przegaliński E, et al. Pol J Pharmacol Pharm. 1986 Jul-Aug;38(4):377-84.
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