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Nefazodone hydrochloride
CAS No. 82752-99-6
Nefazodone hydrochloride( BMY 13754 | MJ13754-1 )
Catalog No. M16074 CAS No. 82752-99-6
Nefazodone hydrochloride is an antidepressant drug.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 67 | In Stock |
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| 5MG | 37 | In Stock |
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| 10MG | 61 | In Stock |
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| 25MG | 117 | In Stock |
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| 50MG | 212 | In Stock |
|
| 100MG | 319 | In Stock |
|
| 200MG | 462 | In Stock |
|
| 500MG | 759 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameNefazodone hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionNefazodone hydrochloride is an antidepressant drug.
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DescriptionNefazodone hydrochloride is an antidepressant drug.(In Vitro):Nefazodone hydrochloride (BMY-13754) is a phenylpiperazine antidepressant with a mechanism of action that is distinct from those of other currently available drugs. Nefazodone hydrochloride potently and selectively blocks postsynaptic serotonin (5-hydroxytryptamine; 5-HT) 5-HT2A receptors and moderately inhibits serotonin and noradrenaline (norepinephrine) reuptake. Nefazodone hydrochloride is also an inhibitor of the hepatic P-450 isoenzyme CYP3A4.
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In VitroNefazodone hydrochloride (BMY-13754) is a phenylpiperazine antidepressant with a mechanism of action that is distinct from those of other currently available drugs. Nefazodone hydrochloride potently and selectively blocks postsynaptic serotonin (5-hydroxytryptamine; 5-HT) 5-HT2A receptors and moderately inhibits serotonin and noradrenaline (norepinephrine) reuptake. Nefazodone hydrochloride is also an inhibitor of the hepatic P-450 isoenzyme CYP3A4.
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In Vivo——
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SynonymsBMY 13754 | MJ13754-1
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor5-HT
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Research AreaNeurological Disease
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Indication——
Chemical Information
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CAS Number82752-99-6
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Formula Weight506.47
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Molecular FormulaC25H33Cl2N5O2
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Purity>98% (HPLC)
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SolubilityDMSO: ~11?mg/mL at?60?°C
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SMILESO=C1N(CCCN2CCN(C3=CC=CC(Cl)=C3)CC2)N=C(CC)N1CCOC4=CC=CC=C4.[H]Cl
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Chemical Name2-(3-(4-(3-chlorophenyl)piperazin-1-yl)propyl)-5-ethyl-4-(2-phenoxyethyl)-2,4-dihydro-3H-1,2,4-triazol-3-one hydrochloride
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Bengi Uslu, et al. Analytica Chimica Acta Volume 462, Issue 1, 26 June 2002, Pages 49–57
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