Cart
sales@molnova.com
Apatinib
CAS No. 811803-05-1
Apatinib( YN968D1 )
Catalog No. M16035 CAS No. 811803-05-1
Apatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 76 | In Stock |
|
| 5MG | 108 | In Stock |
|
| 10MG | 137 | In Stock |
|
| 25MG | 233 | In Stock |
|
| 50MG | 350 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameApatinib
-
NoteResearch use only, not for human use.
-
Brief DescriptionApatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
-
DescriptionApatinib is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.
-
In Vitro——
-
In Vivo——
-
SynonymsYN968D1
-
PathwayAngiogenesis
-
Targetc-Kit
-
Recptorc-Kit| RET| c-Src| VEGFR2
-
Research AreaCancer
-
Indication——
Chemical Information
-
CAS Number811803-05-1
-
Formula Weight397.48
-
Molecular FormulaC24H23N5O
-
Purity>98% (HPLC)
-
SolubilityDMSO: 22 mg/mL (44.57 mM)
-
SMILESCS(O)(=O)=O.O=C(NC1=CC=C(C=C1)C1(CCCC1)C#N)C1=C(NCC2=CC=NC=C2)N=CC=C1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Tian S, et al. Y Sci, 2011, 102(7), 1374-1380.
molnova catalog
related products
-
Sitravatinib
A novel, broad spectrum small molecule inhibitor that blocks a wide array of RTKs known to be amplified/overexpressed in sarcomas, including c-Kit, PDGFRβ, PDGFRα, c-Met, and Axl (IC50=1.5-30 nM).
-
RGB-286638 free base
RGB-286638 free base is a novel CDK inhibitor.
-
Famitinib
Famitinib (SHR1020) is a structural analogue of sunitinib, novel and potent multi-targeted RTK inhibitor.
