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GSK 214096
CAS No. 716354-87-9
GSK 214096( GSK214096 | GSK-214096 )
Catalog No. M15739 CAS No. 716354-87-9
A potent, selective CCR5 antagonist and HIV-1 entry inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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| 100MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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Biological Information
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Product NameGSK 214096
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective CCR5 antagonist and HIV-1 entry inhibitor.
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DescriptionA potent, selective CCR5 antagonist and HIV-1 entry inhibitor.
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In Vitro——
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In Vivo——
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SynonymsGSK214096 | GSK-214096
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PathwayGPCR/G Protein
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TargetChemokine Receptor
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RecptorChemokine Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number716354-87-9
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Formula Weight754.787
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Molecular FormulaC39H46Cl2FN5O3S
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameN-(tert-butyl)-2,4-dichloro-3-(4-(3-fluorophenyl)-4-(2-((1R,3r,5S)-3-(2-methyl-1H-benzo[d]imidazol-1-yl)-8-azabicyclo[3.2.1]octan-8-yl)ethyl)piperidine-1-carbonyl)benzenesulfonamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kazmierski WM, et al. ACS Med Chem Lett. 2014 Oct 28;5(12):1296-9.
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