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GSK 163929
CAS No. 716354-04-0
GSK 163929( GSK163929 | GSK-163929 )
Catalog No. M15738 CAS No. 716354-04-0
A potent, selective CCR5 antagonist and HIV-1 entry inhibitor with pIC50 of 8.37 and 8.46 in HOS and PBL assays, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameGSK 163929
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NoteResearch use only, not for human use.
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Brief DescriptionA potent, selective CCR5 antagonist and HIV-1 entry inhibitor with pIC50 of 8.37 and 8.46 in HOS and PBL assays, respectively.
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DescriptionA potent, selective CCR5 antagonist and HIV-1 entry inhibitor with pIC50 of 8.37 and 8.46 in HOS and PBL assays, respectively.
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In Vitro——
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In Vivo——
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SynonymsGSK163929 | GSK-163929
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PathwayGPCR/G Protein
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TargetChemokine Receptor
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RecptorChemokine Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number716354-04-0
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Formula Weight696.255
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Molecular FormulaC36H40ClF2N5O3S
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name4-chloro-2-fluoro-5-(4-(3-fluorophenyl)-4-(2-((1R,3r,5S)-3-(2-methyl-1H-benzo[d]imidazol-1-yl)-8-azabicyclo[3.2.1]octan-8-yl)ethyl)piperidine-1-carbonyl)-N-methylbenzenesulfonamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kazmierski WM, et al. J Med Chem. 2011 Jun 9;54(11):3756-67.
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