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WAY-100635 maleate (b)

CAS No. 634908-75-1

WAY-100635 maleate (b)( WAY 100635 maleate salt | WAY100635 maleate salt )

Catalog No. M15399 CAS No. 634908-75-1

WAY-100635 is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 58 In Stock
10MG 91 In Stock
25MG 154 In Stock
50MG 221 In Stock
100MG 327 In Stock
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Biological Information

  • Product Name
    WAY-100635 maleate (b)
  • Note
    Research use only, not for human use.
  • Brief Description
    WAY-100635 is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor.
  • Description
    WAY-100635 is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor; completely prevents not only the hyperpolarization, with an IC50 of 1.3 nM, but also the decrease in membrane input resistance produced by 5-HT and 5-carboxamidotryptamine with IC50 of 22.5 μM and 50 nM, respectively.Anxiety Phase 1 Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    WAY 100635 maleate salt | WAY100635 maleate salt
  • Pathway
    GPCR/G Protein
  • Target
    5-HT Receptor
  • Recptor
    5-HT1A
  • Research Area
    Neurological Disease
  • Indication
    Anxiety

Chemical Information

  • CAS Number
    634908-75-1
  • Formula Weight
    538.6352
  • Molecular Formula
    C29H38N4O6
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 34 mg/mL
  • SMILES
    COC1=CC=CC=C1N2CCN(CC2)CCN(C3=CC=CC=N3)C(=O)C4CCCCC4.C(=CC(=O)O)C(=O)O
  • Chemical Name
    Cyclohexanecarboxamide, N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinyl-, (2Z)-2-butenedioate (9CI)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Corradetti R, et al. J Pharmacol Exp Ther. 1996 Aug;278(2):679-88. 2. Fornal CA, et al. J Pharmacol Exp Ther. 1996 Aug;278(2):752-62. 3. García G, et al. Eur J Med Chem. 2014 Oct 6;85:795-806.
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