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C7280948
CAS No. 587850-67-7
C7280948( C7280948 | C-7280948 | C 7280948 )
Catalog No. M15168 CAS No. 587850-67-7
C-7280948 is a PRMT1 inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 36 | In Stock |
|
| 10MG | 58 | In Stock |
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| 25MG | 105 | In Stock |
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| 50MG | 178 | In Stock |
|
| 100MG | 267 | In Stock |
|
| 200MG | 413 | In Stock |
|
| 500MG | 668 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameC7280948
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NoteResearch use only, not for human use.
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Brief DescriptionC-7280948 is a PRMT1 inhibitor.
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DescriptionC-7280948 is a PRMT1 inhibitor.
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In VitroC-7280948 is compound 6a in this article, it against hPRMT1 with an IC50 value of 12.75 μM.Especially arginine methyltransferases also target non-histone protein substrates and are therefore often called protein methyltransferases (PRMTs). The subtype PRMT1 has been linked to the activation of estrogen and androgen receptors and therefore may represent a new treatment option for hormone-dependent cancer.
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In Vivo——
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SynonymsC7280948 | C-7280948 | C 7280948
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorPRMT1
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number587850-67-7
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Formula Weight276.35
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Molecular FormulaC14H16N2O2S
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Purity>98% (HPLC)
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SolubilityDMSO: 10 mM
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SMILESO=S(C1=CC=C(N)C=C1)(NCCC2=CC=CC=C2)=O
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Chemical Name4-amino-N-phenethylbenzenesulfonamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Bissinger EM, et al. Bioorg Med Chem. 2011 Jun 15;19(12):3717-373
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