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Dabigatran ethyl ester
CAS No. 429658-95-7
Dabigatran ethyl ester( Dabigatran ethyl ester | BIBR-951CL | BIBR 951CL | BIBR951CL | UNII-KJ4EH9410G )
Catalog No. M14458 CAS No. 429658-95-7
A reversible and selective, direct thrombin inhibitor (DTI) with Ki value of 4.5 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 32 | In Stock |
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| 5MG | 47 | In Stock |
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| 10MG | 86 | In Stock |
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| 25MG | 158 | In Stock |
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| 50MG | 270 | In Stock |
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| 100MG | 424 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDabigatran ethyl ester
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NoteResearch use only, not for human use.
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Brief DescriptionA reversible and selective, direct thrombin inhibitor (DTI) with Ki value of 4.5 nM.
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DescriptionA reversible and selective, direct thrombin inhibitor (DTI) with Ki value of 4.5 nM; an anticoagulant agent used to prevent stroke with atrial fibrillation.Thrombosis Approved.
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In Vitro——
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In Vivo——
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SynonymsDabigatran ethyl ester | BIBR-951CL | BIBR 951CL | BIBR951CL | UNII-KJ4EH9410G
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PathwayAutophagy
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TargetThrombin
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RecptorThrombin
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Research AreaCardiovascular Disease
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IndicationThrombosis
Chemical Information
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CAS Number429658-95-7
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Formula Weight499.5643
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Molecular FormulaC27H29N7O3
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESO=C(OCC)CCN(C(C1=CC=C2C(N=C(CNC3=CC=C(C(N)=N)C=C3)N2C)=C1)=O)C4=NC=CC=C4
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Chemical Nameβ-Alanine, N-[[2-[[[4-(aminoiminomethyl)phenyl]amino]methyl]-1-methyl-1H-benzimidazol-5-yl]carbonyl]-N-2-pyridinyl-, ethyl ester
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Wienen W, et al. Thromb Haemost. 2007 Jul;98(1):155-62.
2. Kansal AR, et al. Heart. 2012 Apr;98(7):573-8.
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