PPT

CAS No. 263717-53-9

PPT( PPT )

Catalog No. M13809 CAS No. 263717-53-9

An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 92 In Stock
5MG 85 In Stock
10MG 136 In Stock
25MG 264 In Stock
50MG 390 In Stock
100MG 589 In Stock
200MG 827 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    PPT
  • Note
    Research use only, not for human use.
  • Brief Description
    An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
  • Description
    An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
  • In Vitro
    The EC50 of Propyl pyrazole triol for the ERα-dependent response is 140 pM in ERα-U2OS-Luc cells.
  • In Vivo
    ——
  • Synonyms
    PPT
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    GAT
  • Recptor
    GAT
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    263717-53-9
  • Formula Weight
    388.467
  • Molecular Formula
    C24H24N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : ≥ 100 mg/mL (258.77 mM)
  • SMILES
    OC1=CC=C(C2=C(CCC)C(C3=CC=C(O)C=C3)=NN2C4=CC=C(O)C=C4)C=C1
  • Chemical Name
    4,4',4″-(4-propyl-[1H]-pyrazole-1,3,5-triyl)trisphenol

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Yamaura K, et al. Nat Chem Biol. 2016 Oct;12(10):822-30.
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