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PPT

CAS No. 263717-53-9

PPT( PPT )

Catalog No. M13809 CAS No. 263717-53-9

An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 80 In Stock
10MG 129 In Stock
25MG 251 In Stock
50MG 447 In Stock
100MG 669 In Stock
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Biological Information

  • Product Name
    PPT
  • Note
    Research use only, not for human use.
  • Brief Description
    An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
  • Description
    An allosteric GABAA receptor modulator that strongly suppresses GABA-induced chloride currents.
  • In Vitro
    The EC50 of Propyl pyrazole triol for the ERα-dependent response is 140 pM in ERα-U2OS-Luc cells.
  • In Vivo
    ——
  • Synonyms
    PPT
  • Pathway
    Membrane Transporter/Ion Channel
  • Target
    GAT
  • Recptor
    GAT
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    263717-53-9
  • Formula Weight
    388.467
  • Molecular Formula
    C24H24N2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : ≥ 100 mg/mL (258.77 mM)
  • SMILES
    OC1=CC=C(C2=C(CCC)C(C3=CC=C(O)C=C3)=NN2C4=CC=C(O)C=C4)C=C1
  • Chemical Name
    4,4',4″-(4-propyl-[1H]-pyrazole-1,3,5-triyl)trisphenol

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Yamaura K, et al. Nat Chem Biol. 2016 Oct;12(10):822-30.
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