AL082D06

CAS No. 256925-03-8

AL082D06( AL082D06 | AL-082D06 | AL 082D06 | D-06 )

Catalog No. M13775 CAS No. 256925-03-8

AL 082D06(D-06) is the first selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 46 In Stock
5MG 41 In Stock
10MG 73 In Stock
25MG 150 In Stock
50MG 252 In Stock
100MG 335 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    AL082D06
  • Note
    Research use only, not for human use.
  • Brief Description
    AL 082D06(D-06) is the first selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM.
  • Description
    AL 082D06(D-06) is the first selective, nonsteroidal glucocorticoid receptor (GR) antagonist with Ki of 210 nM, exhibits excellent selectivity against AR, PR, MR and ER(Ki > 10 uM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    AL082D06 | AL-082D06 | AL 082D06 | D-06
  • Pathway
    Endocrinology/Hormones
  • Target
    GR
  • Recptor
    Glucocorticoid Receptor
  • Research Area
    Endocrinology
  • Indication
    ——

Chemical Information

  • CAS Number
    256925-03-8
  • Formula Weight
    409.91
  • Molecular Formula
    C23H24ClN3O2
  • Purity
    >98% (HPLC)
  • Solubility
    Soluble in DMSO
  • SMILES
    CN(C)C1=CC=C(C(C2=CC=C(N(C)C)C=C2)C3=CC([N+]([O-])=O)=CC=C3Cl)C=C1
  • Chemical Name
    4,4'-((2-chloro-5-nitrophenyl)methylene)bis(N,N-dimethylaniline)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Avenant C, et al. Mol Cell Endocrinol. 2010 Oct 7;327(1-2):72-88.
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