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CARM1 inhibitor 9
CAS No. 2180931-09-1
CARM1 inhibitor 9( —— )
Catalog No. M13481 CAS No. 2180931-09-1
CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameCARM1 inhibitor 9
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NoteResearch use only, not for human use.
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Brief DescriptionCARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM.
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DescriptionCARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM; displays 20-fold selective for CARM1 over PRMT6 and highly selective over PRMT1, PRMT3, PRMT8 as well as PRMT5 and PRMT7; CARM1 inhibitor 9 is a useful tool for studying the role of CARM1 in health and disease.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorHMTase
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Research Area——
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Indication——
Chemical Information
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CAS Number2180931-09-1
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Formula Weight326.282
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Molecular FormulaC15H24BrN3
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical NameN-(3-bromobenzyl)-1-(2-(methylamino)ethyl)piperidin-4-amine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kaniskan Hü, et al. Medchemcomm. 2016 Sep 1;7(9):1793-1796.
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