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PDE6δ inhibitor 8
CAS No. 2088485-36-1
PDE6δ inhibitor 8( —— )
Catalog No. M13259 CAS No. 2088485-36-1
A novel selective small molecule inhibitor of PDE6δ/KRas interaction with Kd of 358 pM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NamePDE6δ inhibitor 8
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NoteResearch use only, not for human use.
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Brief DescriptionA novel selective small molecule inhibitor of PDE6δ/KRas interaction with Kd of 358 pM.
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DescriptionA novel selective small molecule inhibitor of PDE6δ/KRas interaction with Kd of 358 pM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMAPK/ERK Signaling
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TargetRas
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RecptorRas
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Research Area——
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Indication——
Chemical Information
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CAS Number2088485-36-1
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Formula Weight675.256
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Molecular FormulaC32H39ClN4O6S2
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Purity>98% (HPLC)
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Solubility——
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SMILES——
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Chemical Name2-amino-4-(((4-(N-(4-chlorobenzyl)-N-cyclopentylsulfamoyl)-N-(piperidin-4-ylmethyl)phenyl)sulfonamido)methyl)benzoic acid
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Martín-Gago P, et al. Angew Chem Int Ed Engl. 2017 Feb 20;56(9):2423-2428.
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