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CPI-203
CAS No. 202591-23-9
CPI-203( —— )
Catalog No. M13155 CAS No. 202591-23-9
CPI-203 is a potent BET bromodomain inhibitor with IC50 of 37 nM for BRD4.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 29 | In Stock |
|
| 5MG | 29 | In Stock |
|
| 10MG | 43 | In Stock |
|
| 25MG | 68 | In Stock |
|
| 50MG | 124 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCPI-203
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NoteResearch use only, not for human use.
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Brief DescriptionCPI-203 is a potent BET bromodomain inhibitor with IC50 of 37 nM for BRD4.
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DescriptionCPI-203 is a potent BET bromodomain inhibitor with IC50 of 37 nM for BRD4.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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RecptorBRD4
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Research Area——
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Indication——
Chemical Information
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CAS Number202591-23-9
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Formula Weight399.9
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Molecular FormulaC19H18ClN5OS
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Purity>98% (HPLC)
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SolubilityDMSO: 200 mM
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SMILESCC1=C(C)C2=C(S1)N1C(C)=NN=C1C(CC(N)=O)N=C2C1=CC=C(Cl)C=C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Devaiah BN, et al. Proc natl Acad Sci U S A. 2012, 109(18), 6927-6932.
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