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SGC-2085
CAS No. 1821908-48-8
SGC-2085( SGC2085 | SGC 2085 )
Catalog No. M12811 CAS No. 1821908-48-8
SGC-2085 is a potent, selective protein arginine methyltransferase PRMT4 (CARM1) inhibitor with IC50 of 50 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 155 | In Stock |
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| 2MG | 116 | In Stock |
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| 5MG | 227 | In Stock |
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| 10MG | 341 | In Stock |
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| 25MG | 563 | In Stock |
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| 50MG | 803 | In Stock |
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| 100MG | 1107 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSGC-2085
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NoteResearch use only, not for human use.
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Brief DescriptionSGC-2085 is a potent, selective protein arginine methyltransferase PRMT4 (CARM1) inhibitor with IC50 of 50 nM.
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DescriptionSGC-2085 is a potent, selective protein arginine methyltransferase PRMT4 (CARM1) inhibitor with IC50 of 50 nM, displays >100-fold selectivity over other PRMTs (PRMT6 IC50=5.3 uM); also shows complete selectivity against a panel of 21 human protein methyltransferases.
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In Vitro——
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In Vivo——
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SynonymsSGC2085 | SGC 2085
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PathwayChromatin/Epigenetic
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TargetHMTase
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RecptorCARM1
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1821908-48-8
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Formula Weight312.4061
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Molecular FormulaC19H24N2O2
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 32 mg/mL
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SMILESCC1=CC(=CC(=C1)OC2=C(C=C(C=C2)CNC(=O)C(C)N)C)C
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Chemical NamePropanamide, 2-amino-N-[[4-(3,5-dimethylphenoxy)-3-methylphenyl]methyl]-, (2S)-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ferreira de Freitas R, et al. J Med Chem. 2016 Jul 28;59(14):6838-47.
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